Patent · US Expired

Process for the manufacture of iohexol

US7541494B2 · kind B2 · utility

0Cited by
3References
17Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 3, 2006
Grant dateJun 2, 2009
Priority date
Expiry dateMar 3, 2026

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C231/08
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

A process for the production of iohexol comprises alkylating 5-Acetamido-N,N′-bis(2,3-dihydroxypropyl)-2,4,6-triiodoisophthalamide using 2(2-methoxy-ethoxy)-ethanol as solvent in the presence of a base, and optionally isolating crude iohexol from the reaction mixture. Preferably, the alkylating agent is 1-chloro-2,3 propanediol and the base is an alkali metal hydroxide such as sodium hydroxide or potassium hydroxide.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.