Patent · US Active

Dipeptidyl peptidase-IV inhibitors

US7553861B2 · kind B2 · utility

0Cited by
88References
6Claims
0Family size

Assignee

Inventors

Key dates

Filing dateApr 21, 2006
Grant dateJun 30, 2009
Priority date
Expiry dateJan 3, 2028

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D495/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates generally to pyrrolidine and thiazolidine DPP-IV inhibitor compounds. The present invention also provides synthetic methods for preparation of such compounds, methods of inhibiting DPP-IV using such compounds and pharmaceutical formulations containing them for treatment of DPP-IV mediated diseases, in particular, Type-2 diabetes.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.