Patent · US Expired

Prodrugs of selective androgen receptor modulators and methods of use thereof

US7595402B2 · kind B2 · utility

3Cited by
18References
11Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 16, 2004
Grant dateSep 29, 2009
Priority date
Expiry dateFeb 8, 2026

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C235/24
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides prodrugs of selective androgen receptor modulators (SARMs), and their use in treating or reducing the incidence of osteoporosis, a variety of hormone-related conditions, conditions associated with Androgen Decline in Aging Male (ADAM); conditions associated with Androgen Decline in Female (ADIF), and muscular wasting conditions, obesity, dry eye conditions, and prostate cancer. The prodrugs are also useful in oral androgen replacement therapy and male contraception.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.