Stable hydrate of a muscarinic receptor antagonist
US7696357B2 · kind B2 · utility
Assignee
Inventors
Key dates
| Filing date | Mar 17, 2008 |
| Grant date | Apr 13, 2010 |
| Priority date | — |
| Expiry date | Mar 17, 2028 |
Classification
- Technology area (CPC A)Human Necessities
- CPC primaryA61P43/00
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
A stable solid hydrate of a muscarinic receptor antagonist is useful in the treatment of irritable bowel syndrome, diverticular disease, oesophageal achalasia, chronic obstructive airways disease, over active bladder (including symptoms of incontinence, urge and frequency), urinary incontinence, neurogenic urinary urgency or pollakiuria, treatment of bladder functional disorder, urinary leakage, painful or difficult urination caused by neurogenic bladder, spastic or hypertonic bladder, dysfunctional bladder syndrome, gastrointestinal disorders including gastrointestinal hyperactivity, and relaxing effect on intestinal smooth muscle cells.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.