Patent · US Active

Prodrugs of 5-amino-3-(3′-deoxy-β-D-ribofuranosyl)-thiazolo[4,5-d]pyrimidin-2,7-dione

US7709448B2 · kind B2 · utility

11Cited by
22References
8Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 21, 2007
Grant dateMay 4, 2010
Priority date
Expiry dateJun 27, 2027

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention is directed to 5-amino-3-(3′-deoxy-β-D-ribofuranosyl)-thiazolo[4,5-d]pyrimidin-2,7-dione prodrugs, whose metabolized parent compound has immunomodulatory activity. The invention also relates to the therapeutic use of such prodrugs and pharmaceutical compositions thereof in treating disease states associated with abnormal cell growth, such as cancer.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.