Patent · US Active

2-aminoaryloxazole compounds as tyrosine kinase inhibitors

US7718676B2 · kind B2 · utility

29Cited by
4References
17Claims
0Family size

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Inventors

Key dates

Filing dateOct 22, 2004
Grant dateMay 18, 2010
Priority date
Expiry dateNov 25, 2026

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D413/14
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to novel compounds selected from 2-aminoaryloxazoles of formula I that selectively modulate, regulate, and/or inhibit signal transduction mediated by certain native and/or mutant tyrosine kinases implicated in a variety of human and animal diseases such as cell proliferative, metabolic, allergic, and degenerative disorders. More particularly, these compounds are potent and selective c-kit, bcr-abl, FGFR3 and/or Flt-3 inhibitors.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.