Patent · US Active

Multi-arm cyclic or cubic siloxane-based formulations for drug delivery

US7745547B1 · kind B1 · utility

39Cited by
3References
20Claims
0Family size

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Key dates

Filing dateAug 7, 2006
Grant dateJun 29, 2010
Priority date
Expiry dateDec 13, 2028

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC08L2203/02
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides multi-arm siloxane-based molecules suitable for use as a drug delivery vehicle comprising a central core molecule that comprises a cyclic or cubic siloxane, and a plurality of arms attached to the central core molecule, wherein each arm comprises an organic moiety. The multi-arm siloxane-based molecules described herein are suitable for encapsulation of a therapeutic agent. The invention further includes pharmaceutical compositions comprising the claimed multi-arm siloxane-based molecules and an encapsulated therapeutic agent in combination with a pharmaceutically acceptable carrier. Methods of making and using the multi-arm siloxane-based molecules are also provided.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.