Substituted piperidine compounds and methods of their use
US7767814B2 · kind B2 · utility
3Cited by
12References
62Claims
0Family size
Assignee
Inventors
Key dates
| Filing date | May 25, 2006 |
| Grant date | Aug 3, 2010 |
| Priority date | — |
| Expiry date | Aug 27, 2028 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D221/06
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
Certain 4-aryl-piperidine compounds, including N-substituted 9β-substituted-5-(3-substituted-phenyl)morphans and N-substituted octahydro-4a-(3-hydroxyphenyl)-10a-methyl-benzo[g]isoquinolines, pharmaceutical compositions, and methods of their use, inter alia, as opioid antagonists are disclosed.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.