Patent · US Active

IRE-1α inhibitors

US7858666B2 · kind B2 · utility

12Cited by
119References
24Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 9, 2008
Grant dateDec 28, 2010
Priority date
Expiry dateJun 17, 2028

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02A50/30
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds which directly inhibit IRE-1α activity in vitro, prodrugs, and pharmaceutically acceptable salts thereof. Such compounds and prodrugs are useful for treating diseases associated with the unfolded protein response and can be used as single agents or in combination therapies.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.