Patent · US Active

Capped pyrazinoylguanidine sodium channel blockers

US7868010B2 · kind B2 · utility

36Cited by
25References
15Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 17, 2008
Grant dateJan 11, 2011
Priority date
Expiry dateMar 17, 2028

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D473/16
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention relates to substituted pyrazinoylguanidine compounds. These compounds are useful as sodium channel blockers, and may be effective in treating a variety of conditions including chronic bronchitis and cystic fibrosis.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.