Patent · US Active

Fused tricyclic compounds as serine-threonine protein kinase and PARP modulators

US7956064B2 · kind B2 · utility

20Cited by
1References
14Claims
0Family size

Assignee

Inventors

Key dates

Filing dateAug 31, 2007
Grant dateJun 7, 2011
Priority date
Expiry dateOct 5, 2029

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D513/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention relates in part to fused tricyclic compounds having certain biological activities that include, but are not limited to, inhibiting cell proliferation, modulating protein kinase activity and modulating polymerase activity. The fused tricyclic compounds of the invention can modulate casein kinase (CK) activity and/or poly(ADP-ribose)polymerase (PARP) activity. The invention also relates in part to methods for using such fused tricyclic compounds.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.