Patent · US Active

Indole amide derivatives as EP4 receptor antagonists

US7968578B2 · kind B2 · utility

2Cited by
1References
14Claims
0Family size

Assignee

Inventors

Key dates

Filing dateApr 23, 2007
Grant dateJun 28, 2011
Priority date
Expiry dateJul 24, 2027

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D249/18
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention is directed to indole amide derivatives as EP4 receptor antagonists useful for the treatment of EP4 mediated diseases or conditions, such as acute and chronic pain, osteoarthritis, rheumatoid arthritis and cancer. Pharmaceutical compositions and methods of use are also included.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.