Patent · US Active

Process for the preparation of 6-alpha-hydroxy-N-alkylated opiates

US7985858B2 · kind B2 · utility

7Cited by
15References
21Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 2, 2008
Grant dateJul 26, 2011
Priority date
Expiry dateMay 9, 2029

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02P20/55
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention is directed to the conversion of a 6-keto morphinan to a 6-alpha-hydroxy morphinan in the presence of a ruthenium, rhodium, or iridium asymmetric catalyst and a hydrogen source.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.