Patent · US Active

Purinones and 1H-imidazopyridinones as PKC-theta inhibitors

US7989459B2 · kind B2 · utility

4Cited by
11References
19Claims
0Family size

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Key dates

Filing dateFeb 2, 2007
Grant dateAug 2, 2011
Priority date
Expiry dateNov 18, 2028

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P37/06
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A chemical genus of purinones and 1H-imidazopyridinones, which are useful as PKCθ. inhibitors, and their methods of use are disclosed. The genus is represented by the formula I: A representative example is:

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.