Pyridyl benzoxazine derivatives, pharmaceutical composition comprising the same, and use thereof
US8026235B1 · kind B1 · utility
1Cited by
0References
13Claims
0Family size
Assignee
Inventors
Key dates
| Filing date | Oct 21, 2010 |
| Grant date | Sep 27, 2011 |
| Priority date | — |
| Expiry date | Oct 21, 2030 |
Classification
- Technology area (CPC A)Human Necessities
- CPC primaryA61P43/00
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
Discloses is a benzoxazine benzimidazole derivative, represented by Chemical Formula 1, functioning as an antagonist to the vanilloid receptor-1, a pharmaceutical composition comprising the same, and the use thereof. The benzoxazine benzimidazole derivative can be useful for preventing or treating a disease associated with antagonistic activity of vanilloid receptor-1, without hyperthermia:wherein, R1, R2, R3, R4 and R5 are as defined in the specification.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.