Patent · US Expired

Fused compounds that inhibit vanilloid subtype 1 (VR1) receptor

US8026256B2 · kind B2 · utility

9Cited by
3References
6Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 26, 2005
Grant dateSep 27, 2011
Priority date
Expiry dateOct 26, 2025

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D403/12
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds of formula (I)are novel VR1 antagonists that are useful in treating pain, inflammatory thermal hyperalgesia, urinary incontinence, or bladder overactivity.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.