Antagonists of the TRPV1 receptor and uses thereof
US8030504B2 · kind B2 · utility
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9Claims
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Assignee
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Key dates
| Filing date | Dec 12, 2007 |
| Grant date | Oct 4, 2011 |
| Priority date | — |
| Expiry date | Jan 21, 2030 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D311/74
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
The present application is directed to compounds that are TRPV1 antagonists and have formula (I)wherein variables Ar1, L1, R1, R2, R3, R4, R5, Y1, Y2, and Y3, are as defined in the description, which are useful for treating disorders caused by or exacerbated by vanilloid receptor activity.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.