Patent · US Active

Indole, azaindole and related heterocyclic N-substituted piperazine derivatives

US8039486B2 · kind B2 · utility

2Cited by
14References
11Claims
0Family size

Assignee

Inventors

Key dates

Filing dateFeb 8, 2008
Grant dateOct 18, 2011
Priority date
Expiry dateAug 19, 2030

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D491/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

This invention provides compounds of Formula I, including pharmaceutically acceptable salts thereof, having drug and bio-affecting properties, their pharmaceutical compositions and method of use. These compounds possess unique antiviral activity, whether used alone or in combination with other antivirals, antiinfectives, immunomodulators or HIV entry inhibitors. More particularly, the present invention relates to the treatment of HIV and AIDS. The compounds of Formula I have the formulawherein:

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.