9-(piperazinylalkyl) carbazoles as bax-modulators
US8053436B1 · kind B1 · utility
3Cited by
2References
20Claims
0Family size
Assignee
Inventors
Key dates
| Filing date | Oct 18, 2000 |
| Grant date | Nov 8, 2011 |
| Priority date | — |
| Expiry date | May 7, 2024 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D209/86
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
The present invention is related to piperazine derivatives of carbazole of formula (I) notably for use as pharmaceutically active compounds, as well as to pharmaceutical formulations containing such piperazine derivatives of carbazole. Said piperazine derivatives of carbazole are efficient modulators, in particular efficient inhibitors, of the Bax function and/or activation. The present invention is furthermore related to novel piperazine derivatives of carbazole as well as methods of their preparation.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.