Patent · US Active

Production of rosuvastatin calcium salt

US8063213B2 · kind B2 · utility

1Cited by
28References
13Claims
0Family size

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Inventors

Key dates

Filing dateJun 3, 2004
Grant dateNov 22, 2011
Priority date
Expiry dateApr 8, 2027

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P9/10
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

An improved process for the manufacture of (E)-7-[4-(4-flurophenyl)-6-isopropyl-2-[methyl(methylsulfony)amino]pyrimidin-5-yl](3R,5S)-3,5-dihydroxyhept-6-enoic acid calcium salt, Formula (1), which is useful for the production of a pharmaceutical useful in the treatment of, inter alia, hypercholesterolemia, hyperlipoproteinemia and atherosclerosis, is described.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.