Patent · US Active

Crystalline pharmaceutical and methods of preparation and use thereof

US8080562B2 · kind B2 · utility

32Cited by
56References
21Claims
0Family size

Assignee

Inventors

Key dates

Filing dateApr 15, 2009
Grant dateDec 20, 2011
Priority date
Expiry dateJul 8, 2030

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K47/183
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Novel crystalline polymorphic forms, Forms A, B, C, D, and E of a compound of Formula I, which has been found to be a potent inhibitor of LFA-1, are disclosed. Methods of preparation and uses thereof in the treatment of LFA-1 mediated diseases are also disclosed in this invention.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.