Patent · US Active

Pharmaceutical formulation containing a biguanide and a thiazolidinedione derivative

US8084058B2 · kind B2 · utility

1Cited by
50References
4Claims
0Family size

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Key dates

Filing dateMar 30, 2005
Grant dateDec 27, 2011
Priority date
Expiry dateMar 6, 2028

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K45/06
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A pharmaceutical dosage form comprising a controlled release component comprising an antihyperglycemic drug in combination with a second component comprising a thiazolidinedione derivative and a disintegrating agent is herein disclosed and described. The dosage formulation exhibits a significant increase in bioavailability of the thiazolidinedione derivative component compared to conventional immediate release dosage forms containing only a thiazolidinedione derivative.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.