Patent · US Active

TGR5 modulators and methods of use thereof

US8114862B2 · kind B2 · utility

7Cited by
13References
9Claims
0Family size

Assignee

Inventor

Key dates

Filing dateNov 19, 2009
Grant dateFeb 14, 2012
Priority date
Expiry dateJan 2, 2030

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07J41/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention relates to compounds of Formula A:or a salt, solvate, hydrate, or prodrug thereof. The compounds of Formula A are TGR5 modulators useful for the treatment of various diseases, including metabolic disease, inflammatory disease, liver disease, autoimmune disease, cardiac disease, kidney disease, cancer, and gastrointestinal disease.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.