Patent · US Active

Processes for intermediates for macrocyclic compounds

US8129561B2 · kind B2 · utility

13Cited by
95References
28Claims
0Family size

Assignee

Inventors

Key dates

Filing dateNov 19, 2008
Grant dateMar 6, 2012
Priority date
Expiry dateJan 8, 2029

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07K5/0827
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention is directed to novel macrocyclic compounds of formula (I) and their pharmaceutically acceptable salts, hydrates or solvates:wherein R1, R2, R3, R4, R5, R6, n1, m, p Z1, Z2, and Z3 are as describe in the specification. The invention also relates to compounds of formula (I) which are antagonists of the motilin receptor and are useful in the treatment of disorders associated with this receptor and with or with motility dysfunction.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.