Patent · US Active

Substituted picolinamides as MAO-B inhibitors useful for treating obesity

US8138209B2 · kind B2 · utility

4Cited by
8References
20Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 12, 2006
Grant dateMar 20, 2012
Priority date
Expiry dateOct 10, 2030

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07F9/6512
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The invention provides novel compounds of formula I:that are monoamine oxidase-B inhibitors, which can be useful in treating obesity, diabetes, and/or cardiometabolic disorders (e.g., hypertension, dyslipidemias, high blood pressure, and insulin resistance).

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.