Patent · US Active

Aurora kinase inhibitors from an encoded small molecule library

US8138338B2 · kind B2 · utility

0Cited by
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13Claims
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Assignee

Inventor

Key dates

Filing dateJul 27, 2007
Grant dateMar 20, 2012
Priority date
Expiry dateJul 27, 2027

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D401/12
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides, at least in part, compounds of formula (I): or a pharmaceutically acceptable salt thereof, wherein Z1, Z2, Z3, R1, x, y, R2, R3, R4a, R4b, R5, R6 and R7 are described herein, as well as methods for their identification, their preparation, pharmaceutical compositions containing them, and their use as Aurora A kinase inhibitors in treatment, e.g., of cancer and other proliferative disorders.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.