Patent · US Active

Inhibitors of protein kinases

US8138339B2 · kind B2 · utility

49Cited by
36References
19Claims
0Family size

Assignee

Inventors

Key dates

Filing dateApr 16, 2009
Grant dateMar 20, 2012
Priority date
Expiry dateJul 11, 2029

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D413/14
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention is directed to 2-cycloalkylamino-4-arylamino-benzamide compounds of formula I pharmaceutically acceptable salts thereof which are inhibitors of syk and/or JAK kinase. The present invention is also directed to intermediates used in making such compounds, the preparation of such a compound, pharmaceutical compositions containing such a compound, methods of inhibition syk and/or JAK kinase activity, and methods to prevent or treat a number of conditions mediated at least in part by syk and/or JAK kinase activity, such as cardiovascular disease, inflammatory disease, autoimmune disease and cell proliferative disorder.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.