Patent · US Active

Quinoline derivatives as PI3 kinase inhibitors

US8138347B2 · kind B2 · utility

147Cited by
6References
4Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 16, 2008
Grant dateMar 20, 2012
Priority date
Expiry dateJun 19, 2030

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D498/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Invented is a method of inhibiting the activity/function of PI3 kinases using quinoline derivatives. Also invented is a method of treating one or more disease states selected from: autoimmune disorders, inflammatory diseases, cardiovascular diseases, neurodegenerative diseases, allergy, asthma, pancreatitis, multiorgan failure, kidney diseases, platelet aggregation, cancer, sperm motility, transplantation rejection, graft rejection and lung injuries by the administration of quinoline derivatives.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.