Patent · US Active

Substituted pyridone derivative

US8158652B2 · kind B2 · utility

0Cited by
3References
7Claims
0Family size

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Inventors

Key dates

Filing dateNov 30, 2005
Grant dateApr 17, 2012
Priority date
Expiry dateNov 22, 2028

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds of a formula (I)[wherein, A represents formula (III-1)R3 is a hydrogen, lower alkyl et al; m is 0 or 1; R1 is a hydrogen atom, halogen atom et al, R2 is a hydrogen et al; p is 0 to 4; X is a carbon atom or nitrogen atom; and X1 to X4 is a lower alkyl et al], or pharmaceutical acceptable salts thereof. These have a potency antagonistic to binding to histamine H3 receptor, or have a potency inhibiting the constant activity of histamine H3 receptor, and are useful in the therapy of obesity, diabetes et al.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.