Patent · US Active

Methods of using substituted isoxazolo pyridinones as dissociated glucocorticoids

US8173670B2 · kind B2 · utility

2Cited by
3References
9Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJan 13, 2010
Grant dateMay 8, 2012
Priority date
Expiry dateJan 13, 2030

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P37/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A method for treating a subject having an inflammatory or auto-immune disease with a substituted isoxazolo pyridinone. Also, a method for administering a substituted isoxazolo pyridinone to a cell to retain or increase glucocorticoid receptor transrepression activity with only minimal glucocorticoid receptor transactivation activity.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.