Patent · US Active

Quinazolinones as inhibitors of human phosphatidylinositol 3-kinase delta

US8207153B2 · kind B2 · utility

43Cited by
41References
6Claims
0Family size

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Key dates

Filing dateMar 25, 2010
Grant dateJun 26, 2012
Priority date
Expiry dateJun 3, 2030

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds that inhibit P13Kδ activity, including compounds that selectively inhibit P13Kδ activity, are disclosed. Methods of inhibiting phosphatidylinositol 3-kinase delta isoform (P13Kδ) activity, and methods of treating diseases, such as disorders of immunity and inflammation in which P13Kδ plays a role in leukocyte function, using the compounds also are disclosed.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.