Patent · US Active

Compound having affinity for amyloid

US8207189B2 · kind B2 · utility

1Cited by
10References
16Claims
0Family size

Assignee

Inventors

Key dates

Filing dateAug 16, 2007
Grant dateJun 26, 2012
Priority date
Expiry dateJul 14, 2028

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P25/28
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A compound represented by the following formula or a salt thereof:wherein each of A1, A2, A3 and A4 independently represents a carbon or nitrogen, R1 is a radioactive halogen substituent, R2 is a group selected from the group consisting of hydrogen, a hydroxyl group, a methoxy group, a carboxyl group, an amino group, an N-methylamino group, an N,N-dimethylamino group and a cyano group, and p is an integer of 0 to 2, provided at least one of A1, A2, A3 and A4 represents a carbon, and R1 binds to a carbon represented by A1, A2, A3 or A4, is effective as an image diagnosis probe targeting amyloid. A diagnostic agent for Alzheimer's disease contains the compound.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.