Patent · US Active

Cannabinoid receptor antagonists/inverse agonists useful for treating metabolic disorders, including obesity and diabetes

US8217038B2 · kind B2 · utility

1Cited by
8References
14Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 7, 2010
Grant dateJul 10, 2012
Priority date
Expiry dateOct 7, 2030

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D413/12
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides novel pyrazolines that are useful as cannabinoid receptor blockers and pharmaceutical compositions thereof and methods of using the same for treating obesity, diabetes, inflammatory disorders, cardiometabolic disorders, hepatic disorders, and/or cancers.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.