Patent · US Active

Liquid phase peptide synthesis of KL-4 pulmonary surfactant

US8217142B2 · kind B2 · utility

0Cited by
12References
2Claims
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Assignee

Inventors

Key dates

Filing dateSep 30, 2008
Grant dateJul 10, 2012
Priority date
Expiry dateDec 7, 2028

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K38/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention relates to improved liquid phase processes for the preparation of the 21 residue protein component, (Lys-Leu4)4-Lys, of the pulmonary surfactant KL-4. These process are amenable to large scale synthesis and one process employs a method of saponifying an ester which reduces the inherent racemization of the α-carbon.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.