Patent · US Active

Heteroaryloxy quinazoline derivative

US8232284B2 · kind B2 · utility

1Cited by
1References
15Claims
0Family size

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Inventors

Key dates

Filing dateNov 10, 2008
Grant dateJul 31, 2012
Priority date
Expiry dateApr 6, 2029

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D513/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Disclosed are compounds of the following formula and their pharmaceutically-acceptable salts, which have an effect of glucokinase activation and are useful in the field of medicines for treatment for diabetes, obesity, etc.(wherein ring A represents a pyrazolyl group optionally having a lower alkyl group, etc.; ring B represents a heteroaryl group; R represents a lower alkyl group, etc.; R1 represents a group of a formula:(wherein R11 and R12 each independently represent a hydrogen atom, etc.; m indicates an integer of from 2 to 6), etc.;R2 represents a lower alkyl group, etc.; r indicates an integer of from 0 to 3; k indicates an integer of from 0 to 4).

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.