Patent · US Active

Pyrazine derivatives as ENAC blockers

US8236808B2 · kind B2 · utility

20Cited by
1References
8Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 8, 2009
Grant dateAug 7, 2012
Priority date
Expiry dateJun 8, 2029

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D403/12
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A compound of Formula Ior a hydrate or solvate thereof, where R1, R2, R3, R4, R5, R6, R7, R8, R9, and R10 have the meanings as indicated in the specification, is useful for treating diseases which respond to the blockade of the epithelial sodium channel. Pharmaceutical compositions that contain the compounds and processes for preparing the compounds are also described.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.