Patent · US Active

Substituted N-phenyl-5-phenyl-pyrazolin-3-yl amides as cannabinoid receptor antagonists/inverse agonists useful for treating obesity

US8236821B2 · kind B2 · utility

1Cited by
0References
12Claims
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Assignee

Inventors

Key dates

Filing dateMay 19, 2009
Grant dateAug 7, 2012
Priority date
Expiry dateJul 5, 2030

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07F9/65031
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention provides novel pyrazolines that are useful as cannabinoid receptor antagonists/inverse agonists and pharmaceutical compositions thereof and methods of using the same for treating obesity, diabetes, dyslipidemias, cardiovascular disorders, hepatic disorders, and a combination thereof.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.