Patent · US Active

Bicycloamine derivatives

US8252810B2 · kind B2 · utility

6Cited by
0References
9Claims
0Family size

Assignee

Inventors

Key dates

Filing dateFeb 9, 2009
Grant dateAug 28, 2012
Priority date
Expiry dateNov 6, 2030

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D519/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds represented by formula (I) and pharmaceutically acceptable salts thereof have excellent sodium channel inhibitory action and are useful as therapeutic agents and analgesics for various kinds of neuralgia, neuropathy, epilepsy, insomnia, premature ejaculation and the like.wherein Q represents ethylene, etc., R1, R2 and R3 represent hydrogen, etc., X1 represents C1-6 alkylene, etc., X2 represents C1-6 alkylene, etc., A1 represents a 5- to 6-membered heterocyclic group, etc., and A2 represents C6-14 aryl, etc.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.