Patent · US Active

Antagonists of the bradykinin B1 receptor

US8278280B2 · kind B2 · utility

0Cited by
19References
14Claims
0Family size

Assignee

Inventors

Key dates

Filing dateApr 8, 2008
Grant dateOct 2, 2012
Priority date
Expiry dateJun 2, 2031

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07K7/18
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to composition of matter involving bradykinin B1 receptor antagonist peptides conjugated to a multivalent vehicle, including peptides conjugated to multivalent PEG. These compositions can be used as therapeutics or prophylactics against diseases or conditions, such as inflammation or pain, linked to the bradykinin B1 receptor.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.