Patent · US Active

Imidazolo-, oxazolo-, and thiazolopyrimidine modulators of TRPV1

US8288397B2 · kind B2 · utility

1Cited by
1References
20Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 16, 2008
Grant dateOct 16, 2012
Priority date
Expiry dateFeb 28, 2031

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D498/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Certain TRPV1-modulating imidazolo-, oxazolo-, and thiazolopyrimdine compounds are described. The compounds may be used in pharmaceutical compositions and methods for treating disease states, disorders, and conditions mediated by TRPV1 activity, such as pain, arthritis, itch, cough, asthma, or inflammatory bowel disease.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.