Patent · US Active

Method for producing thiazole compound

US8304558B2 · kind B2 · utility

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7References
5Claims
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Assignee

Inventors

Key dates

Filing dateJan 11, 2007
Grant dateNov 6, 2012
Priority date
Expiry dateJun 18, 2027

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D277/32
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Disclosed is a simple and advantageous method for producing a thiazole compound, which method is suitable for commercial-scale implementation. In this method, a thiazole compound is produced by a reaction between 2-halogeno-allylisothiocyanate and sulfuryl chloride generating a large amount of heat, while suppressing decrease in the yield of the thiazole compound. Specifically disclosed is a method for producing 2-chloro-5-chloromethylthiazole represented by the formula (1):This method is characterized in that sulfuryl chloride is added to and reacted with 2-halogeno-allylisothiocyanate represented by the formula (2):wherein Hal represents chlorine or bromine, while blowing a gas inactive to the reaction into the reaction liquid.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.