Patent · US Active

Cephalosporin derivatives and pharmaceutical compositions thereof

US8329684B2 · kind B2 · utility

5Cited by
0References
19Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 8, 2012
Grant dateDec 11, 2012
Priority date
Expiry dateMay 8, 2032

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02A50/30
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention relates to novel cephalosporin derivatives represented by Chemical Formula 1.Wherein, X, Y, L, R1, and R2 are as same as defined in the description of the invention. The present invention also relates to pharmaceutical antibiotic compositions comprising a novel celphalosporin derivative represented by Chemical Formula 1, a prodrug thereof, a hydrate thereof, a solvate thereof, an isomer thereof, or a pharmaceutically acceptable salt thereof as an effective ingredient. Compounds of the present invention are effective ingredients for the broad spectrum of antibiotic resistance, exhibit low toxicity, particularly in Gram-negative bacteria, which can be useful with strong antimicrobial activity.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.