Patent · US Active

N-containing heterocyclic compounds

US8354408B2 · kind B2 · utility

8Cited by
1References
11Claims
0Family size

Assignee

Inventors

Key dates

Filing dateNov 14, 2008
Grant dateJan 15, 2013
Priority date
Expiry dateNov 14, 2028

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D513/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to N-containing heterocyclic compounds that are inhibitors of protein kinases including JAK kinases. In particular, the compounds are selective for JAK1, JAK2, JAK3 or TYK2 kinases and combinations thereof such as JAK1 and JAK2. The kinase inhibitors can be used in the treatment of kinase associated diseases such as immunological and inflammatory diseases including organ transplants; hyperproliferative diseases including cancer and myeloproliferative diseases; viral diseases; metabolic diseases; and vascular diseases.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.