Patent · US Active

Crystalline pharmaceutical and methods of preparation and use thereof

US8367701B2 · kind B2 · utility

29Cited by
62References
41Claims
0Family size

Assignee

Inventors

Key dates

Filing dateNov 4, 2011
Grant dateFeb 5, 2013
Priority date
Expiry dateNov 4, 2031

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K47/183
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Novel crystalline polymorphic forms, Forms A, B, C, D, and E of a compound of Formula I, which has been found to be a potent inhibitor of LFA-1, are disclosed. Methods of preparation and uses thereof in the treatment of LFA-1 mediated diseases are also disclosed in this invention.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.