Patent · US Active

Trisubstituted thiophenes that modulate intracellular calcium

US8372991B2 · kind B2 · utility

2Cited by
3References
14Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 17, 2011
Grant dateFeb 12, 2013
Priority date
Expiry dateMar 17, 2031

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D495/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Described herein are compounds of Formula (I):wherein A, J, Z, X, R1 and R4 are defined herein, and pharmaceutical compositions containing such compounds, which modulate the activity of store-operated calcium (SOC) channels. Also described herein are methods of using such SOC channel modulators, alone and in combination with other compounds, for treating diseases or conditions that would benefit from inhibition of SOC channel activity.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.