Patent · US Active

Controlled release carvedilol compositions

US8449914B2 · kind B2 · utility

11Cited by
21References
32Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 13, 2008
Grant dateMay 28, 2013
Priority date
Expiry dateOct 18, 2028

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K31/403
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A controlled release pharmaceutical composition for oral use comprising carvedilol. The composition releases carvedilol after oral administration to a mammal, including a human, in such a manner that a prolonged residence of carvedilol is obtained in the circulatory system compared with the known compositions of carvedilol. Furthermore, a composition according to the present invention makes available to the body a suitable plasma concentration of one or both of the enantiomeric species, namely R(+) and/or S(−) carvedilol for obtaining the desired therapeutic effect.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.