Patent · US Active

Formulation

US8466139B2 · kind B2 · utility

15Cited by
16References
20Claims
0Family size

Assignee

Inventors

Key dates

Filing dateSep 4, 2012
Grant dateJun 18, 2013
Priority date
Expiry dateSep 4, 2032

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K47/44
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention relates to a novel sustained release pharmaceutical formulation adapted for administration by injection containing the compound 7α-[9-(4,4,5,5,5-pentafluoropentylsulphinyl)nonyl]oestra-1,3,5(10)-triene-3,17β-diol, more particularly to a formulation adapted for administration by injection containing the compound 7α-[9-(4,4,5,5,5-pentafluoropentylsulphinyl)nonyl]oestra-1,3,5(10)-triene-3,17β-diol in solution in a ricinoleate vehicle which additionally comprises at least one alcohol and a non-aqueous ester solvent which is miscible in the ricinoleate vehicle.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.