Patent · US Active

Methods for isolating crystalline form I of 5-azacytidine

US8481715B2 · kind B2 · utility

2Cited by
25References
12Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 5, 2012
Grant dateJul 9, 2013
Priority date
Expiry dateJun 5, 2032

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07H19/12
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The invention includes methods for isolating crystalline Form I of 5-azacytidine substantially free of other forms, wherein 5-azacytidine is represented by the formula:The invention also includes pharmaceutical compositions comprising Form I of 5-azacytidine.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.