Patent · US Active

Bis-aryl amide compounds and methods of use

US8492404B2 · kind B2 · utility

10Cited by
8References
7Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 26, 2010
Grant dateJul 23, 2013
Priority date
Expiry dateNov 3, 2030

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D495/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention comprises a new class of compounds useful for the prophylaxis and treatment of protein kinase mediated diseases, including autoimmune disease and inflammation. In one embodiment, the compounds have a general Formula Iwherein A1, A2, A3, A4, L, R1, R2 and R3 are defined herein. The invention also comprises pharmaceutical compositions including one or more compounds of the present invention, methods of use such as treatment of Lck and/or c-Kit kinase mediated diseases by administering the compounds of the invention, or compositions including one or more compounds of the invention, and intermediates and processes useful for the preparation of compounds of the present invention.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.