Patent · US Expired

Controlled release formulation of erythromycin derivatives

US8507000B2 · kind B2 · utility

4Cited by
9References
47Claims
0Family size

Assignee

Inventor

Key dates

Filing dateMay 6, 2004
Grant dateAug 13, 2013
Priority date
Expiry dateMay 6, 2024

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K9/2866
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention is directed to a controlled release formulation in tablet form comprising a pharmaceutically effective amount of an erythromycin derivative and a lubricating effective amount of a lubricant in the absence of material selected from the group consisting of alginic acid or salts thereof or hydrophilic sustained release polymers in amounts effective to retard the release of the erythromycin derivatives in the pharmaceutical composition. It is also directed to a method for facilitating the release of erythromycin derivative from a pharmaceutical composition comprising a therapeutically effective amount of a lubricating effective amount of a lubricant said method comprising adding to said composition an release promoter in tablet disintegrating effective amounts to facilitate the release of the erythromycin derivative from the tablet.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.